3'-AROYL-4'-HYDROXY-1'-(2-HYDROXYMETHYLPHENYL)-2H,4H-SPIRO[1,4-BENZOTHIAZINE-2,2'-PYRROLE]-3,5'(1'H)-DIONES, HAVING ANALGESIC ACTIVITY Russian patent published in 2020 - IPC C07D513/10 A61K31/5415 A61P29/00 

Abstract RU 2714511 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to 3'-aroyl-4'-hydroxy-1'-(2-hydroxymethylphenyl)-2H,4H-spiro[1,4-benzothiazine-2,2'-pyrrole]-3,5'(1'H)-dions of general formula:

having analgesic activity.

EFFECT: obtaining novel compounds of the spiro[1,4-benzothiazine-2,2'-pyrrol]diones, which can be used in pharmacology as having analgesic activity.

1 cl, 4 ex, 1 tbl

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RU 2 714 511 C1

Authors

Maslivets Anna Andreevna

Maslivets Andrej Nikolaevich

Makhmudov Ramiz Ragibovich

Tretyakov Nikita Alekseevich

Dates

2020-02-18Published

2019-09-06Filed