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2 471 798

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IPC

C07D487/04(2006-01-01)

A61K31/4985(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2011132175/04, 2011-07-29

(24)

Start date

2011-07-29

(22)

Actual filing date

2011-07-29

(45)

Published

2013-01-10

(72)

Inventor

Mashevskaja Irina VladimirovnaKislina Lalita ViktorovnaMakhmudov Ramiz RagibovichMaslivets Andrej Nikolaevich

(73)

Holder

Gosudarstvennoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet"

3-AROYL-2-(2-ARYLHYDRAZONO)PYRROLO [1,2-a] QUINOXALINE,4-(2H,5H)DIONES POSSESSING ANALGESIC ACTIVITY Russian patent published in 2013 - IPC C07D487/04 A61K31/4985 A61P29/00

Abstract RU 2471798 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to 3-aroyl-2-arylhydrazonopyrrolo[1,2-a]quinozaline-1,4(2H,5H)-diones of formula:

Ar=Ph, R=Me, R¹=H (a); Ar=4-MeC₆H₄ R=Me, R¹=H (b); Ar=Ph, R=H, R¹=COOH (c).

EFFECT: there are produced new compounds possessing analgesic activity that makes them being suggested to be used in medicine as drugs with the analgesic properties.

1 cl, 3 tbl, 4 ex

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RU 2 471 798 C1

Authors

Mashevskaja Irina Vladimirovna

Kislina Lalita Viktorovna

Makhmudov Ramiz Ragibovich

Maslivets Andrej Nikolaevich

Dates

2013-01-10—Published

2011-07-29—Filed