(Z)-4-ARYL-N-[2-(2-HYDROXYMETHYL)PHENYL]-2,4-DIOXO-3-[3-OXO-3,4-DIHYDROQUINOXALINE-2(1N)-YLIDENE]BUTANAMIDES, HAVING ANALGESIC ACTIVITY Russian patent published in 2020 - IPC C07D241/44 C07D241/38 A61K31/498 A61P29/00 

Abstract RU 2722178 C1

FIELD: chemistry.

SUBSTANCE: invention relates to (Z)-4-aryl-N-[2-(2-hydroxymethyl)phenyl]-2,4-dioxo-3-[3-oxo-3,4-dihydroquinoxalin-2(1H)-ylidene]butanamides of general formula given below, where Ar = 4-ClC6H4, 4-CH3C6H4, 4-CH3OC6H4.

EFFECT: technical result is obtaining novel compounds which can be used in medicine as drugs with analgesic properties.

1 cl, 4 ex, 1 tbl

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RU 2 722 178 C1

Authors

Maslivets Anna Andreevna

Maslivets Andrej Nikolaevich

Makhmudov Ramiz Ragibovich

Tretyakov Nikita Alekseevich

Dates

2020-05-28Published

2019-09-06Filed