FIELD: pharmaceuticals.
SUBSTANCE: invention relates to specific compounds specified in claim 1, as well as to a compound having general formula given below, where R4 is selected from hydrogen, halogen and C1-C6 alkyl; and Y is a group having formula given below, where L is absent, each R313 is independently selected from H, halogen and C1-C6 alkyl and R" is selected from H and C1-C6 alkyl or its pharmaceutically acceptable salts. Declared compounds inhibit tryptophan-2,3-dioxygenase (TDO) or indolamine-2,3-dioxygenase (IDO). Invention also relates to pharmaceutical compositions based on said compounds. .
EFFECT: disclosed is a pharmaceutical compound.
6 cl, 2 dwg, 3 tbl, 2 ex
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Authors
Dates
2020-04-17—Published
2015-11-02—Filed