IMIDAZO[1,2-A]PYRIDINE DERIVATIVES, METHODS FOR PRODUCTION THEREOF AND USE THEREOF Russian patent published in 2020 - IPC C07D471/04 C07D403/06 A61K31/437 A61K31/397 A61P1/00 

Abstract RU 2725147 C1

FIELD: chemistry.

SUBSTANCE: present invention relates to an imidazo[1,2-a]pyridine derivative of general formula I, having inhibitory activity on gastric acid secretion, a pharmaceutical composition based thereon, method of treatment and use for treating a disease caused by excessive secretion of gastric acid. In general formula IY1, Y2 and Y3, each, independently, is H, halogen, straight-chain C1-C6 alkyl, unsubstituted or substituted with R1 or hydroxy; R1 is hydroxy; Y4 represents H, C1-C6 straight chain alkyl or C1-C6 alkoxy; and X is H or halogen.

EFFECT: treatment of the disease caused by excessive secretion of gastric acid.

10 cl, 1 dwg, 4 tbl, 48 ex

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RU 2 725 147 C1

Authors

Kim, Jeongmin

Lee, Hyunho

Chun, Kwangwoo

Park, Chun-Ho

Jang, Eunsung

Park, Yoonsun

Kim, Joseph

Dates

2020-06-30Published

2017-07-04Filed