FIELD: medicine; pharmaceuticals.
SUBSTANCE: invention relates to benzoxazepinoxazolidinones of formula I, pharmaceutical compositions on and base selectively inhibiting PI3Kα mutant form, methods of treating cancer, associated with expression of mutant form PI3Kα.
(I).
EFFECT: obtaining novel compounds suitable for treating cancer associated with expression of mutant form PI3Kα.
23 cl, 21 tbl, 3 dwg
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