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2 734 877

(13)

(51)

IPC

C07D487/04(2006-01-01)

A61K31/519(2006-01-01)

A61P33/02(2006-01-01)

(21) (22)

Application

2018107657, 2016-08-03

(24)

Start date

2016-08-03

(22)

Actual filing date

2016-08-03

(45)

Published

2020-10-23

(72)

Inventor

Brand, StephenDodd, Peter GeorgeKo, Eun JungMarco Martin, MariaMiles, Timothy JamesSandberg, Lars HenrikThomas, Michael GeorgeThompson, Stephen

(73)

Holder

Glaxosmithkline Intellectual Property Development LimitedUniversity Of Dundee

COMPOUNDS Russian patent published in 2020 - IPC C07D487/04 A61K31/519 A61P33/02

Abstract RU 2734877 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention refers to compounds of formula (I), pharmaceutical compositions, use and method of treatment.

EFFECT: obtaining novel compounds having anti-parasitic activity mediated by Trypanosoma cruzi or Leishmania donovani, and suitable for treating diseases such as Chagas disease, human African trypanosomiasis, African animal trypanosomiasis and leishmaniasis, particularly visceral leishmaniasis.

13 cl, 57 ex

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RU 2 734 877 C2

Authors

Brand, Stephen

Dodd, Peter George

Ko, Eun Jung

Marco Martin, Maria

Miles, Timothy James

Sandberg, Lars Henrik

Thomas, Michael George

Thompson, Stephen

Dates

2020-10-23—Published

2016-08-03—Filed