TRANSGLUTAMINASE 2 (TG2) INHIBITORS Russian patent published in 2022 - IPC C07D401/06 C07D401/14 C07D403/06 C07D405/14 C07D413/06 C07D413/14 C07D417/06 C07D417/14 C07D471/04 C07D473/30 C07D473/34 C07D487/04 A61K31/4439 A61K31/444 A61K31/497 A61K31/501 A61K31/506 A61K31/52 A61P1/16 A61P11/00 A61P13/12 A61P25/28 A61P27/02 A61P35/00 A61P43/00 C07K5/62 C07K5/78 

Abstract RU 2781370 C2

FIELD: pharmaceutical chemistry.

SUBSTANCE: group of inventions relates to pharmaceutical chemistry and includes specific compounds specified in the claims, a pharmaceutical composition based on them, a method for the treatment of a disease or a disorder mediated by transglutaminase 2, and the use of compounds in the production of a drug.

EFFECT: compounds, which inhibit transglutaminase 2 (TG2).

22 cl, 1 tbl, 109 ex

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RU 2 781 370 C2

Authors

Campbell, David

Chapman, Justin

Cheung, Mui, H.

Diraimondo, Thomas, R.

Duron, Sergio, G.

Dates

2022-10-11Published

2019-08-09Filed