FIELD: pharmaceuticals.
SUBSTANCE: invention relates to dipharmacophoric compounds of nootropic-analgesic action of the formula (1), where the R-radicals of acid NSAIDs, such as ibuprofen, diclofenac, indomethacin, niflumic acid, mefenamic acid, ketoprofen, dexketoprofen, naproxen, diflunisal, sublet, ketorolbene, tolmetin, etodolac, flufenamic acid, meclofenamic acid, tolfenamic acid, dexindoprofen.
EFFECT: new dipharmacophore compounds have been obtained, which exhibit both analgesic and nootropic effects, which allows using the proposed compounds with an analgesic effect at the same time to enhance human cognitive actions in conditions of complicated human activity.
(1)
1 cl, 22 ex, 11 dwg
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Authors
Dates
2021-03-11—Published
2020-04-10—Filed