FIELD: organic chemistry.
SUBSTANCE: present invention relates to the field of organic chemistry, namely, to the compound of the formula (I) or its pharmacologically acceptable salt, tautomer or deuterated analog:
(I),
in which R1 is a cyano, halogen, or (C1-C3)alkyl; and X is absent. Also proposed is a pharmaceutical composition for modulating the bromodomain, a method for modulating the bromodomain, a method for treating the subject, a compound suitable for obtaining a compound of formula (I), a method for obtaining a compound of the formula (I).
EFFECT: proposed are new organic compounds that modulate bromodomain.
17 cl, 2 dwg, 9 tbl, 7 ex
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