PHARMACEUTICAL COMPOSITIONS OF SUBSTITUTED QUINAZOLINONES Russian patent published in 2017 - IPC A61K31/517 A61K9/48 A61P3/06 A61P9/00 A61P35/00 

Abstract RU 2640115 C2

FIELD: pharmacology.

SUBSTANCE: composition according to this invention contains an active ingredient selected from a series of substituted quinazolinones and their pharmaceutically acceptable salts, stereoisomers, tautomers or hydrates, and additionally contains approximately 10 wt % to approximately 85 wt % of microcrystalline cellulose; approximately 4.0 wt % of sodium starch glycolate; approximately 0.5 wt % of magnesium stearate; and approximately 2.5 wt % of colloidal silicon dioxide; and prepared for peroral introduction and immediate release.

EFFECT: creation of new compounds that increase the bioavailability of substituted quinazolinones while maintaining stability, possibility of treatment and prevention of the abovementioned diseases.

15 cl, 1 tbl, 1 ex

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RU 2 640 115 C2

Authors

Shinoj Narmada R.

Dates

2017-12-26Published

2012-10-31Filed