CRYSTAL OF PYRROLOPYRIMIDINE FOR OBTAINING JAK INHIBITOR Russian patent published in 2021 - IPC C07D487/04 A61K31/519 A61K31/5377 A61P35/00 

Abstract RU 2746045 C2

FIELD: chemistry.

SUBSTANCE: invention relates to crystal A and crystal B of acetonitrile of the compound represented by formula I, pharmaceutical compositions based on them, their use for the preparation of a medicament for the treatment or prevention of Janus kinase-mediated disease.

EFFECT: crystal A and crystal B of the compound represented by formula I have high purity and good stability and are suitable for industrial production.

13 cl, 6 dwg, 6 tbl, 5 ex

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RU 2 746 045 C2

Authors

Chzhou Chzhou

Chzhan Ajmin

Chzhan Sitsyuan

Yao Khuadun

Dates

2021-04-06Published

2017-06-15Filed