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2 761 950

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IPC

A61K31/499(2006-01-01)

A61K31/506(2006-01-01)

A61P31/14(2006-01-01)

(21) (22)

Application

2020140398, 2020-12-08

(24)

Start date

2020-12-08

(22)

Actual filing date

2020-12-08

(45)

Published

2021-12-14

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Inventor

Makarov Vadim AlbertovichRyabova Olga BorisovnaMonakhova Natalya SergeevnaChepur Sergej ViktorovichPluzhnikov Nikolaj NikolaevichMyasnikov Vadim AleksandrovichYudin Mikhail AnatolevichTyunin Mikhail AleksandrovichIlinskij Nikita Sergeevich

(73)

Holder

Federalnoe Gosudarstvennoe Uchrezhdenie Issledovatelskij Tsentr Osnovy Biotekhnologii» Rossijskoj Akademii Nauk»Obshchestvo S Ogranichennoj Otvetstvennostyu Innovatsionnoe Predpriyatie Pdstp»

DERIVATIVES OF DI(DIAZONIADISPIRO[5.2.5.2]HEXADECANE)-5-NITROPYRIMIDINE AND THEIR USE FOR TREATMENT OF CORONAVIRUS INFECTIONS, IN PARTICULAR CAUSED BY SARS-COV-2 VIRUS Russian patent published in 2021 - IPC A61K31/499 A61K31/506 A61P31/14

Abstract RU 2761950 C1

FIELD: medicine.

SUBSTANCE: invention relates to the field of medicine, namely, it is aimed at treating or preventing coronavirus infection in humans or animals caused by the SARS-Cov-2 virus by using a compound of general formula 1, where R is CH₃, or its hydrochloride salt, dihydrochloride salt or hexahydrate dihydrochloride.

EFFECT: high antiviral activity against coronavirus infection in humans or animals caused by the SARS-Cov-2 virus.

4 cl, 6 tbl, 9 ex

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RU 2 761 950 C1

Authors

Makarov Vadim Albertovich

Ryabova Olga Borisovna

Monakhova Natalya Sergeevna

Chepur Sergej Viktorovich

Pluzhnikov Nikolaj Nikolaevich

Myasnikov Vadim Aleksandrovich

Yudin Mikhail Anatolevich

Tyunin Mikhail Aleksandrovich

Ilinskij Nikita Sergeevich

Dates

2021-12-14—Published

2020-12-08—Filed