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2 771 031

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IPC

C07D227/10(2006-01-01)

A61K31/402(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2021121412, 2021-07-19

(24)

Start date

2021-07-19

(22)

Actual filing date

2021-07-19

(45)

Published

2022-04-25

(72)

Inventor

Rubtsov Aleksandr EvgenevichMakhmudov Ramiz Ragibovich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Natsionalnyj Issledovatelskij Universitet"

ETHYL ETHER (5 E)-2-AMINO-5-[2-(4-METHYLPHENYL)-2-HYDROXYETHYLIDENE]-1-(3-NITROPHENYL)-4-OXO-1H-4,5-DIHYDROPYRROL-3-CARBOXYLIC ACID, WITH ANTINOCICEPTIVE ACTIVITY Russian patent published in 2022 - IPC C07D227/10 A61K31/402 A61P29/00

Abstract RU 2771031 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to the use of biologically active substances of class 2-aminopyrroles, namely, ethyl ether (5E)-2-amino-5-[2-(4-methylphenyl)-2-oxoethylidene]-1-(3-nitrophenyl)-4-oxo-1H-4,5-dihydropyrrol-3-carboxylic acid, general formula

, as analgesics.

EFFECT: compound ethyl ether (5E)-2-amino-5-[2-(4-methylphenyl)-2-oxoethylidene]-1-(3-nitrophenyl)-4-oxo-1H-4,5-dihydropyrrol-3-carboxylic acid has pronounced analgesic activity, as well as low toxicity.

1 cl, 1 tbl

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RU 2 771 031 C1

Authors

Rubtsov Aleksandr Evgenevich

Makhmudov Ramiz Ragibovich

Dates

2022-04-25—Published

2021-07-19—Filed