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2 773 397

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IPC

C07D487/22(2006-01-01)

A61K31/409(2006-01-01)

A61K31/4439(2006-01-01)

(21) (22)

Application

2021133747, 2021-11-18

(24)

Start date

2021-11-18

(22)

Actual filing date

2021-11-18

(45)

Published

2022-06-03

(72)

Inventor

Syrbu Sergej AleksandrovichKiselev Aleksej NikolaevichGubarev Yurij AleksandrovichLebedeva Natalya ShamilevnaSemejkin Aleksandr StanislavovichKojfman Oskar Iosifovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Khimiko-Tekhnologicheskij Universitet"Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Institut Khimii Rastvorov Im. G.A. Krestova Rossijskoj Akademii Nauk Ran)

5-[4-(1,3-BENZOTHIAZOL-2-YL)PHENYL]-10,15,20-TRIS(1-METHYLPYRIDINIUM-3-YL)PORPHYRIN TRIIOODIDE, SHOWING THE BINDING PROPERTY OF THE SARS-CoV-2 VIRUS SPIKE PROTEIN Russian patent published in 2022 - IPC C07D487/22 A61K31/409 A61K31/4439

Abstract RU 2773397 C1

FIELD: chemistry.

SUBSTANCE: invention relates to 5-[4-(1,3-benzothiazol-2-yl)phenyl]-10,15,20-tris(1-methylpyridinium-3-yl)porphyrin triiodide of the formula:

EFFECT: proposed compound exhibits the property of binding to the SARS-CoV-2 spike protein and can be used as the active basis of a drug that has an inhibitory ability against the SARS-CoV-2 spike protein.

1 cl, 3 dwg, 1 tbl, 1 ex

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RU 2 773 397 C1

Authors

Syrbu Sergej Aleksandrovich

Kiselev Aleksej Nikolaevich

Gubarev Yurij Aleksandrovich

Lebedeva Natalya Shamilevna

Semejkin Aleksandr Stanislavovich

Kojfman Oskar Iosifovich

Dates

2022-06-03—Published

2021-11-18—Filed