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2 785 688

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IPC

C07D239/10(2006-01-01)

A61K31/505(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2022118394, 2022-07-06

(24)

Start date

2022-07-06

(22)

Actual filing date

2022-07-06

(45)

Published

2022-12-12

(72)

Inventor

Gein Vladimir LeonidovichZamaraeva Tatiana MikhailovnaRudakova Irina Pavlovna

(73)

Holder

Federalnoe Gosudarstvennoe Biudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Gosudarstvennaia Farmatsevticheskaia Akademiia» Ministerstva Zdravookhraneniia Rossiiskoi Federatsii

USE OF 3,4-DIMETHYL-6-(3-NITROPHENYL)-2-OXO-N-PHENYL-1,2,3,6-TETRAHYDROPYRIMIDINE-5-CARBOXAMIDE AS AGENT WITH ANALGESIC ACTIVITY Russian patent published in 2022 - IPC C07D239/10 A61K31/505 A61P29/00

Abstract RU 2785688 C1

FIELD: pharmaceutics.

SUBSTANCE: invention relates to biologically active compounds. The use of 3,4-dimethyl-6-(3-nitrophenyl)-2-oxo-N-phenyl-1,2,3,6-tetrahydropyrimidine-5-carboxamide of the formula (1) as an agent with analgesic activity is proposed.

EFFECT: detection of high analgesic activity of 3,4-dimethyl-6-(3-nitrophenyl)-2-oxo-N-phenyl-1,2,3,6-tetrahydropyrimidine-5-carboxamide with its low toxicity, which makes it possible to use it as a new analgesic drug.

1 cl, 2 tbl, 2 ex

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RU 2 785 688 C1

Authors

Gein Vladimir Leonidovich

Zamaraeva Tatiana Mikhailovna

Rudakova Irina Pavlovna

Dates

2022-12-12—Published

2022-07-06—Filed