USE OF 5-BENZOYL-4-HYDROXY-N-(4-IODOPHENYL)-6-(4-CHLOROPHENYL)-2-OXOHEXAHYDROPYRIMIDINE-4-CARBOXAMIDE AS AGENT WITH ANALGESIC ACTIVITY Russian patent published in 2024 - IPC A61K31/513 A61P29/00 C07D239/10 

Abstract RU 2811249 C1

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to the use of biologically active compounds of the class N,6-diaryl-5-aroyl-4-hydroxy-2-oxohexahydropyrimidine-4-carboxamides, namely to the use of 5-benzoyl-4-hydroxy-N-(4-iodophenyl)-6-(4-chlorophenyl)-2-oxohexahydropyrimidine-4-carboxamide of formula (1) as an agent having analgesic activity.

EFFECT: analgesic activity of 5-benzoyl-4-hydroxy- N- (4-iodophenyl)-6-(4-chlorophenyl)-2-oxohexahydropyrimidine-4-carboxamide, which can be used in pharmacology and medicine as an analgesic drug, as well as for the synthesis of new heterocyclic systems.

1 cl, 2 tbl, 2 ex

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RU 2 811 249 C1

Authors

Gorgopina Ekaterina Vladimirovna

Zamaraeva Tatiana Mikhailovna

Rudakova Irina Pavlovna

Gein Vladimir Leonidovich

Dates

2024-01-11Published

2023-06-06Filed