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2 790 479

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IPC

C07D513/10(2006-01-01)

A61K31/429(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2022119903, 2022-07-20

(24)

Start date

2022-07-20

(22)

Actual filing date

2022-07-20

(45)

Published

2023-02-21

(72)

Inventor

Maslivets Andrei NikolaevichTretiakov Nikita AlekseevichBalandina Svetlana Iurevna

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Gosudarstvennyi Natsionalnyi Issledovatelskii Universitet»

APPLICATION OF 9-AROYL-8-HYDROXY-6-(2-HYDROXYALKYL)-2-IMINO-1-THIA-3,6-DIAZASPIRO[4,4]NON-8-EN-4,7-DIONES AS AGENTS, WITH ANTIMICROBIAL ACTIVITY Russian patent published in 2023 - IPC C07D513/10 A61K31/429 A61P31/04

Abstract RU 2790479 C1

FIELD: chemistry.

SUBSTANCE: invention relates to the use of 9-aroyl-8-hydroxy-6-(2-hydroxyalkyl)-2-imino-1-thia-3,6-diazaspiro[4,4]non-8-en-4,7-diones of the total formulas

where R¹=Н, R²=Н, Ar=4-СН₃С₆Н₄; R¹=Me, R²=Н, Ar=Ph; R¹=Н, R²=Ph, Ar=4-BrC₆H₄, as antimicrobial agents.

EFFECT: new compounds that can be used in pharmacology as having antimicrobial activity.

1 cl, 1 tbl, 4 ex

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RU 2 790 479 C1

Authors

Maslivets Andrei Nikolaevich

Tretiakov Nikita Alekseevich

Balandina Svetlana Iurevna

Dates

2023-02-21—Published

2022-07-20—Filed