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2 813 484

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IPC

A61K31/4166(2006-01-01)

A61K31/4188(2006-01-01)

A61P31/04(2006-01-01)

C07D487/10(2006-01-01)

(21) (22)

Application

2023106314, 2023-03-17

(24)

Start date

2023-03-17

(22)

Actual filing date

2023-03-17

(45)

Published

2024-02-12

(72)

Inventor

Tretiakov Nikita AlekseevichMaslivets Andrei NikolaevichBalandina Svetlana Iurevna

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Gosudarstvennyi Natsionalnyi Issledovatelskii Universitet»

USE OF 9-AROYL-8-HYDROXY-6-(2-HYDROXYALKYL)-1,3-DIPHENYL-1,3,6-TRIAZASPIRO[4,4]NON-8-ENE-2,4,7-TRIONES AGENTS WITH ANTIMICROBIAL ACTIVITY AGAINST S. AUREUS CULTURE Russian patent published in 2024 - IPC A61K31/4166 A61K31/4188 A61P31/04 C07D487/10

Abstract RU 2813484 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to the use of compounds of formula 4a-b, where R = H, Ar = Ph (a); R = H, Ar = 4-CH₃C₆H₄(b); R = CH₃, Ar = 4-BrC₆H₄ (c), class of triazaspiro[4,4]nonenetriones as agents with antimicrobial activity against S. aureus.

EFFECT: invention provides antimicrobial activity against S. aureus and can find application in pharmacology.

1 cl, 4 ex, 1 tbl

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RU 2 813 484 C1

Authors

Tretiakov Nikita Alekseevich

Maslivets Andrei Nikolaevich

Balandina Svetlana Iurevna

Dates

2024-02-12—Published

2023-03-17—Filed