METHOD FOR PRODUCING 2-[(3R)-3-METHYLMORPHOLIN-4-YL]-4-(1-METHYL-1H-PYRAZOL-5-YL)-8-(1H-PYRAZOL-5-YL)-1,7-NAFTHYRIDINE Russian patent published in 2023 - IPC C07D471/04 

Abstract RU 2802512 C2

FIELD: chemical industry.

SUBSTANCE: invention relates to a method for obtaining 2-[(3R)-3-methylmorpholin-4-yl]-4-(1-methyl-1H-pyrazol-5-yl)-8-(1H-pyrazol-5-yl)-1 ,7-naphthyridine ("compound of formula (I)", as well as intermediate compounds suitable for obtaining compounds of formula (I).

EFFECT: new effective method for obtaining a compound of formula (I) has been developed, which makes it possible to obtain a product with a high yield and purity.

20 cl, 6 dwg, 1 tbl, 7 ex

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Authors

Platzek Johannes

Rubenbauer Philipp

Van Der Haas Hendricus Nicolaas Sebastiaan

Hoogeveen Sonja Elisabeth

Van Oers Matthijs Cornelis Maria

Gieling Reinerus Gerardus

Dekker Jeroen Alexander

Dates

2023-08-30Published

2019-08-22Filed