FIELD: pharmaceuticals.
SUBSTANCE: invention relates to a bifunctional chelator for the production of radiopharmaceuticals including the DOTA chelator with 4-methoxybenzaldehyde of the formula indicated below attached to it through the methylene group. The invention is aimed at solving the problem of possibly more simply and efficiently obtaining a wide range of precursors for radiopharmaceuticals, primarily containing peptides as vectors aimed at targets in the tumor.
EFFECT: production of a bifunctional DOTA chelator for the production of radiopharmaceutical precursors.
1 cl, 4 ex
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Authors
Dates
2023-11-30—Published
2023-04-04—Filed