USE OF 1'-ARYLDISPIRO[CYCLOALKANE-1,3'-AZETIDINE-2',3''-INDOLINE]-2'',4'-DIONES AS ANALGESICS Russian patent published in 2023 - IPC A61K31/397 A61K31/404 A61P29/02 C07D487/10 C07D471/10 

Abstract RU 2809008 C1

FIELD: organic chemistry.

SUBSTANCE: invention relates to the new use of 1'-aryldispiro[cycloalkane-1,3'-azetidine-2',3''-indoline]-2'',4'-diones, expressed by formulas 1a-c as analgesics.

EFFECT: suppression of pain sensitivity provided by compounds of the specified structure 1a-c, which have pronounced analgesic activity.

1 cl, 1 tbl, 4 ex

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RU 2 809 008 C1

Authors

Nikiforova Elena Aleksandrovna

Zverev Dmitrii Pavlovich

Makhmudov Ramiz Ragibovich

Uchuskin Maksim Grigorevich

Mendogralo Elena Iurevna

Makarov Anton Sergeevich

Rubtsov Aleksandr Evgenevich

Sergeeva Serafima Valerevna

Dates

2023-12-05Published

2023-05-03Filed