FIELD: organic chemistry.
SUBSTANCE: invention relates to new biologically active substances of the class of substituted 2-amino-4-dioxobutanoic acids and is intended to reduce pain sensitivity. 4-oxo-4-(thiophen-2-yl)-2-{[4-(4-chlorophenyl)-3-(ethoxycarbonyl)thiophen-2-yl]amino}but-2-enoic acid is used as a medicine with analgesic properties.
EFFECT: use of the invention makes it possible to obtain a compound with high yield, which has pronounced analgesic activity, as well as low toxicity.
1 cl, 1 tbl, 3 ex
| Title |
Year |
Author |
Number |
| APPLICATION OF 2-[(3-(AMINOCARBONIL)-4,5,6,7-TETRAHYDROBENZO[b]THIOPHEN-2-yl)AMINO]-4-OXO-4-(4-CHLOROPHENYL)BUT-2-ENOIC ACID IN AS AN ANTI-INFLAMMATORY DRUG |
2022 |
- Shipilovskikh Sergei Aleksandrovich
- Makhmudov Ramiz Ragibovich
- Rubtsov Aleksandr Evgenevich
|
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2012 |
- Shipilovskikh Sergej Aleksandrovich
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- Makhmudov Ramiz Ragibovich
|
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|
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|
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|
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|
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|
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|
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