(Z)-2-((4-R-5-R-3-(ETHOXYCARBONYL)THIOPHEN-2-YL)AMINO)-4-OXO-4-R-BUT-2-ENE ACIDS, HAVING ANTIMICROBIAL ACTIVITY Russian patent published in 2020 - IPC C07D333/72 C07D333/70 A61K31/381 A61P31/00 

Abstract RU 2722176 C1

FIELD: chemistry.

SUBSTANCE: invention relates to use of (Z)-2-((4-R1-5-R2-3-(ethoxycarbonyl)thiophen-2-yl)amino)-4-oxo-4-R3-but-2-ene acids 1-3 of general formula:

as an antimicrobial agent.

EFFECT: technical result is obtaining compounds having pronounced antimicrobial activity, as well as low toxicity.

1 cl, 1 tbl, 5 ex

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RU 2 722 176 C1

Authors

Shipilovskikh Sergej Aleksandrovich

Rubtsov Aleksandr Evgenevich

Makhmudov Ramiz Ragibovich

Dates

2020-05-28Published

2019-09-06Filed