4-OXO-2-{[4-PHENYL-3-(ETHOXYCARBONYL)THIOPHEN-2-YL]AMINO)}-4-(4-FLUOROPHENYL)BUT-2-ENOIC ACID, HAVING ANTI-INFLAMMATORY ACTIVITY Russian patent published in 2024 - IPC C07D333/38 A61K31/381 A61P29/00 

Abstract RU 2831129 C1

FIELD: organic chemistry.

SUBSTANCE: invention relates to organic chemistry, specifically to 4-oxo-2-{[4-phenyl-3-(ethoxycarbonyl)thiophen-2-yl]amino)}-4-(4-fluorophenyl)but-2-enoic acid (1).

EFFECT: obtaining a compound of formula 1, having pronounced anti-inflammatory activity and low toxicity.

1 cl, 1 tbl, 3 ex

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RU 2 831 129 C1

Authors

Shipilovskikh Sergej Aleksandrovich

Makhmudov Ramiz Ragibovich

Gorbunova Irina Aleksandrovna

Sharaveva Yuliya Olegovna

Dates

2024-12-02Published

2024-04-04Filed