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2 813 896

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IPC

A61K31/443(2006-01-01)

A61P29/00(2006-01-01)

C07D405/04(2006-01-01)

(21) (22)

Application

2023118670, 2023-07-14

(24)

Start date

2023-07-14

(22)

Actual filing date

2023-07-14

(45)

Published

2024-02-19

(72)

Inventor

Bibik Igor ValerevichPokrovskii Mikhail VladimirovichBibik Elena IurevnaKrivokolysko Sergei Gennadievich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Gosudarstvennyi Natsionalnyi Issledovatelskii Universitet"

2-METHYL-N-(2-METHYLPHENYL)-4-(2-FURYL)-5-CYANO-6-({2-[(4-ETHOXYPHENYL)AMINO]-2-OXOETHYL}THIO)-1,4-DIHYDROPYRIDINE-3-CARBOXAMIDE EXHIBITING ANALGESIC PROPERTIES Russian patent published in 2024 - IPC A61K31/443 A61P29/00 C07D405/04

Abstract RU 2813896 C1

FIELD: medicine.

SUBSTANCE: invention relates to medical chemistry and pharmacology, specifically to use of 2-methyl-N-(2-methylphenyl)-4-(2-furyl)-5-cyano-6-({2-[(4-ethoxyphenyl)amino]-2-oxoethyl}thio)-1,4-dihydropyridine-3-carboxamide of formula (I) as an analgesic.

EFFECT: providing more pronounced analgesic action of the compound of formula (I) compared to such a preparation as sodium metamizole.

1 cl, 1 tbl, 2 ex

(I)

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RU 2 813 896 C1

Authors

Bibik Igor Valerevich

Pokrovskii Mikhail Vladimirovich

Bibik Elena Iurevna

Krivokolysko Sergei Gennadievich

Dates

2024-02-19—Published

2023-07-14—Filed