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2 840 384

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IPC

C07D405/04(2006-01-01)

A61K31/443(2006-01-01)

A61P29/00(2006-01-01)

(21) (22)

Application

2024122622, 2024-08-07

(24)

Start date

2024-08-07

(22)

Actual filing date

2024-08-07

(45)

Published

2025-05-22

(72)

Inventor

Krivokolysko Sergei GennadievichBibik Elena IurevnaFrolov Konstantin AleksandrovichBocheva Anastasiia Aleksandrovna

(73)

Holder

Federalnoe Gosudarstvennoe Biudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Gosudarstvennyi Meditsinskii Universitet Imeni Sviatitelia Luki» Minzdrava Rossii Vo Lgmu Im. Sviat. Luki Mz Rf)

ALLYL-2-METHYL-6-((2-((4-NITROPHENYL)AMINO)-2-OXYETHYL)THIO)-5-CYANO-4-(FURAN-2-YL)-1,4-DIHYDROPYRIDIN-3-CARBOXYLATE EXHIBITING ANALGESIC PROPERTIES Russian patent published in 2025 - IPC C07D405/04 A61K31/443 A61P29/00

Abstract RU 2840384 C1

FIELD: pharmaceuticals.

SUBSTANCE: invention refers to medical or pharmaceutical chemistry and pharmacology. Disclosed is the use of allyl-2-methyl-6-((2-((4-nitrophenyl)amino)-2-oxyethyl)thio)-5-cyano-4-(furan-2-yl)-1,4-dihydropyridin-3-carboxylate of formula (I), given below, as an analgesic agent.

EFFECT: pronounced analgesic action of the compound of formula (I).

1 cl, 2 tbl, 2 ex

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RU 2 840 384 C1

Authors

Krivokolysko Sergei Gennadievich

Bibik Elena Iurevna

Frolov Konstantin Aleksandrovich

Bocheva Anastasiia Aleksandrovna

Dates

2025-05-22—Published

2024-08-07—Filed