TERPENE-BASED QUATERNARY AMMONIUM COMPOUNDS HAVING ANTIMICROBIAL ACTIVITY Russian patent published in 2024 - IPC C07C233/36 C07C323/41 A61P31/02 A61P31/04 A61P31/10 

Abstract RU 2818914 C1

FIELD: chemistry.

SUBSTANCE: invention relates to novel terpene-based quaternary ammonium compounds of general formula (I), which exhibit antimicrobial activity and can be used in medicine and veterinary science. Values of R1 and R2 are given below.

EFFECT: disclosed are compounds exhibiting antimicrobial activity.

1 cl, 1 dwg, 13 ex

No. R1 R2 No. R1 R2 I1 (CH2)10CH3
(+)-myrtenol residue
I7 (CH2)12CH3
(+)-myrtenol residue
I2 (CH2)10CH3
(-)-myrtenol residue
I8 (CH2)12CH3
(-)-myrtenol residue
I3 (CH2)10CH3
(-)-perilla alcohol residue
I9 (CH2)12CH3
(-)-perilla alcohol residue
I4 (CH2)10CH3
(+)-ethylthioborneol residue
I10 (CH2)12CH3
(+)-ethylthioborneol residue
I5 (CH2)10CH3
(-)-citronellol residue
I11 (CH2)12CH3
(-)-citronellol residue
I6 (CH2)10CH3
geraniol residue
I12 (CH2)12CH3
geraniol residue

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Authors

Nikitina Liliia Evgenevna

Pavelev Roman Sergeevich

Gilfanov Ilmir Rafisovich

Lisovskaia Svetlana Anatolevna

Kaiumov Airat Rashitovich

Trizna Elena Iurevna

Ostolopovskaia Olga Viacheslavovna

Dates

2024-05-07Published

2023-12-05Filed