HETEROCYCLIC COMPOUNDS, METHODS FOR PRODUCTION AND USE THEREOF Russian patent published in 2024 - IPC C07D471/04 C07D519/00 A61K31/519 A61P35/00 

Abstract RU 2828748 C2

FIELD: medicine; pharmaceutics.

SUBSTANCE: invention relates to heterocyclic compounds, specifically to a compound or a pharmaceutically acceptable salt thereof, where the compound is

Invention also relates to a pharmaceutical composition, a method of inhibiting the mutant KRAS G12C protein in a cell and a method of treating cancer associated with the G12C mutation in KRAS, based on said compounds.

EFFECT: obtaining alternative compounds for treating cancer associated with G12C mutation in KRAS.

9 cl, 6 dwg, 4 tbl, 23 ex

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RU 2 828 748 C2

Authors

Dai Xing

Wang Yaolin

Jiang Yueheng

Liu Yanqin

Shi Zhe

Wang Zhenwu

Tao Liangshan

Han Zixing

Niu Haotao

Weng Jifang

Dates

2024-10-17Published

2020-05-20Filed