HETEROCYCLIC COMPOUNDS FOR TYK2 ACTIVITY INHIBITION Russian patent published in 2025 - IPC C07D403/12 A61K31/501 A61P29/00 

Abstract RU 2833524 C1

FIELD: chemistry.

SUBSTANCE: invention relates to compounds selected from:

or their pharmaceutically acceptable salts, which are selective binding agents for JH2 TYK2 and exhibit a significant inhibitory effect on the physiological function of TYK2.

EFFECT: obtaining novel compounds which selectively bind JH2 TYK2 and exhibit a significant inhibitory effect on the physiological function of TYK2, as well as having excellent pharmacokinetic properties in vivo.

4 cl, 2 dwg, 4 tbl, 14 ex

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RU 2 833 524 C1

Authors

Chen, Xiangyang

Pang, Yucheng

Dates

2025-01-23Published

2021-03-09Filed