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2 834 046

(13)

(51)

IPC

C07D231/38(2006-01-01)

A61K31/415(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2024120598, 2024-07-22

(24)

Start date

2024-07-22

(22)

Actual filing date

2024-07-22

(45)

Published

2025-02-03

(72)

Inventor

Meshcheriakova Anna ArkadevnaKonstantinova Ekaterina AndreevnaBurygin Gennadii LeonidovichSorokin Vitalii Viktorovich

(73)

Holder

Federalnoe Gosudarstvennoe Biudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Natsionalnyi Issledovatelskii Gosudarstvennyi Universitet Imeni N.G. Chernyshevskogo"

5-AMINO-1-(2,4-DINITROPHENYL)-3-(2-METHOXYPHENYL)-1H-PYRAZOLE-4-CARBONITRILE, HAVING ANTIMICROBIAL PROPERTIES Russian patent published in 2025 - IPC C07D231/38 A61K31/415 A61P31/04

Abstract RU 2834046 C1

FIELD: chemistry.

SUBSTANCE: invention relates to pharmaceutical chemistry, specifically to 5-amino-1-(2,4-dinitrophenyl)-3-(2-methoxyphenyl)-1H-pyrazole-4-carbonitrile of formula (I) or a pharmaceutically acceptable salt thereof.

EFFECT: compound of formula (I) exhibiting antibacterial activity against gram-negative (Pseudomonas aeruginosa and Escherichia coli) and gram-positive (Staphylococcus aureus) bacteria.

3 cl, 1 tbl

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RU 2 834 046 C1

Authors

Meshcheriakova Anna Arkadevna

Konstantinova Ekaterina Andreevna

Burygin Gennadii Leonidovich

Sorokin Vitalii Viktorovich

Dates

2025-02-03—Published

2024-07-22—Filed