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2 838 320

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(51)

IPC

A61K31/407(2006-01-01)

A61P31/04(2006-01-01)

C07D209/96(2006-01-01)

(21) (22)

Application

2024139901, 2024-12-27

(24)

Start date

2024-07-24

(22)

Actual filing date

2024-12-27

(45)

Published

2025-04-14

(72)

Inventor

Sorokin Vitalii ViktorovichMeshcheriakova Anna ArkadevnaKonstantinova Ekaterina AndreevnaBurygin Gennadii LeonidovichBorisova Svetlana Vasilevna

(73)

Holder

Federalnoe Gosudarstvennoe Biudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Natsionalnyi Issledovatelskii Gosudarstvennyi Universitet Imeni N.G. Chernyshevskogo"

1'-(2,3,4-TRIMETHOXYPHENYL)-2-OXO-5',6',7',7a'-TETRAHYDROSPIRO[INDOLINE-3,3'-PYRROLYSINE]-2',2'(1'H)-DICARBONITRILE, HAVING ANTIMICROBIAL PROPERTIES Russian patent published in 2025 - IPC A61K31/407 A61P31/04 C07D209/96

Abstract RU 2838320 C1

FIELD: pharmaceutical chemistry.

SUBSTANCE: invention discloses use of 1'-(2,3,4-trimethoxyphenyl)-2-oxo-5',6',7',7a'-tetrahydrospiro[indoline-3,3'-pyrrolysine]-2',2'(1'H)-dicarbonitrile of formula (I) or a pharmaceutically acceptable salt thereof as an agent having antimicrobial activity against the bacterium Pseudomonas aeruginosa.

EFFECT: invention provides a wider range of pharmaceutical agents due to a representative of substituted spiropyrrolizide indicarbonitriles.

1 cl, 1 tbl

Similar patents RU2838320C1

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RU 2 838 320 C1

Authors

Sorokin Vitalii Viktorovich

Meshcheriakova Anna Arkadevna

Konstantinova Ekaterina Andreevna

Burygin Gennadii Leonidovich

Borisova Svetlana Vasilevna

Dates

2025-04-14—Published

2024-12-27—Filed