DOSING REGIMEN FOR TREATING A CSF-1R-MODULATED DISEASE Russian patent published in 2025 - IPC A61K31/426 A61K31/4427 A61K31/4439 A61P21/00 A61P35/00 

Abstract RU 2835316 C1

FIELD: pharmaceutics.

SUBSTANCE: invention refers to pharmaceutical industry, namely to a method of treating amyotrophic lateral sclerosis. Method of treating amyotrophic lateral sclerosis in a subject, comprising administering to said subject of 4-((2-(((1R,2R)-2-hydroxycyclohexyl)amino)benzo[d]thiazol-6-yl)oxy)-N-methylpicolinamide or a pharmaceutically acceptable salt thereof for period of 4 days, followed by a period of no administration of 10 days, and in a daily dose of 600 mg/day, 800 mg/day or 1200 mg/day.

EFFECT: use of the invention provides reduced probability of undesirable phenomena, namely reduced probability of AST and ALT level increase.

10 cl, 13 dwg, 10 tbl, 8 ex

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RU 2 835 316 C1

Authors

Jullion, Astrid

Meille, Christophe

Quadt, Cornelia

Roy, Michael John

Wiesmann, Marion

Dates

2025-02-24Published

2021-04-19Filed