FIELD: organic chemistry. SUBSTANCE: the product: sulfur- containing heterocyclic compounds of the formula: wherein A is a benzene ring and may be substituted by 1 or 2 substituents selected from the group consisting of halogen, alkyl, alkoxyl or cycloalkyl; R is hydrogen, alkyl or phenyl; B is carboxyl alkoxycarbonyl or an unsubstituted or substituted amido group; X is hydroxyalkyl or carbonyl; K is 0-1 or 0-2, or salts thereof, are prepared by cyclization of the corresponding benzene A derivative followed optionally by oxidation and/or hydrolysis followed by amidation or hydrolysis followed by amidation and oxidation and optionally by reduction. EFFECT: improved properties of the title compounds. 3 cl, 19 tbl
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DERIVATIVES OF 1,2,4-TRIAZOLE, OPTICALLY INERT OR CONTAINING R- OR S-CONFIGURATION AT C-2 AND C-3 ASYMMETRIC CENTERS, OR THEIR SALTS SHOWING FUNGICIDE ACTIVITY, AND A METHOD OF THEIR SYNTHESIS |
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BENZIMIDAZOLE DERIVATIVES, METHOD OF THEIR SYNTHESIS AND PHARMACEUTICAL COMPOSITION ON THEIR BASIS |
1991 |
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METHOD OF SYNTHESIS OF IMIDAZO-(1,2-B)-PYRIDAZINE OR THEIR SALTS AND IMIDAZO-(1,2-B)-PYRIDAZINE DERIVATIVES OR THEIR SALTS |
1990 |
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1993 |
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METHOD OF SYNTHESIS OF BENZIMIDAZOLE DERIVATIVES OR THEIR SALTS |
1990 |
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HETEROCYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION, METHOD OF ANTAGONISM OF ANGIOTENSIN-II |
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THIENOPYRIMIDINE DERIVATIVES, METHOD FOR THEIR PREPARING, PHARMACEUTICAL COMPOSITION AND METHOD FOR ANTAGONIZATION OF GONADOTROPIN-RELEASING HORMONE |
2000 |
- Furuja Suiti
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OPTICALLY ACTIVE BENZOTHIEPINE DERIVATIVE, METHOD OF ITS SYNTHESIS, ACTIVATORS OF OSTEOGENESIS, METHOD OF ACTIVATION OF OSTEOGENESIS, METHODS OF TREATMENT |
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