FIELD: organic chemistry. SUBSTANCE: products: substituted hexahydrobenz[cd]indoles of the formula (I) showing activity of serotonine function modification. Reagent 1: compound of the formula (II). Reagent 2: CO. Reagent 3: compound of the formula (III). Reaction conditions: heating in the presence of palladium-containing catalyst, for example, (Ph3P)4Pd. Method involves removal of amino-protective group B. Synthesized compounds were used in pharmaceutical industry. EFFECT: improved method of synthesis. 1 tbl
| Title |
Year |
Author |
Number |
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1992 |
- Majkl Ehdvard Flaf[Us]
- Majkl Dzhon Martinelli[Us]
- Dzhon Menert Skauz[Us]
|
RU2073672C1 |
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1992 |
- Richard Nolan Bukher[Us]
- Dehvid Ehrnst Lokhorn[Us]
- Majkl Dzhon Martinelli[Us]
- Charl'Z Dzhonson Pehjdzhet
- Dzhon Menert Skaus[Us]
|
RU2062775C1 |
| METHOD OF SYNTHESIS OF TETRAHYDROBENZ(C,D)INDOLE AGONISTS OF SEROTONIN |
1990 |
- Majkl Ehdvard Flau[Us]
- Mark Mortensen Foreman[Us]
|
RU2007393C1 |
| USE OF 6-HETEROCYCLO-4-AMINO-1,3,4,5-TETRAHYDROBENZ[CD]INDOLE USED IN VOMITING OR NAUSEA AT MOVING, PHARMACEUTICAL COMPOSITION |
1993 |
- Richard Nolan Bukher
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- Dzhon Menert Shos
|
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0 |
|
SU1375128A3 |
| 4-(DI-N-PROPYL)AMINOCARBONYL-1,3,4,5-TETRAHYDROBENZ (CD) INDOLE HIPPURATE AND 4R-AND 4S-ISOMERS THEREOF |
1992 |
- Tomas Dzhozef Kress[Us]
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|
RU2083561C1 |
| PROCESS FOR PREPARING HYPPURATE OF 4-(DI-N-PROPYL) ANINO- 6-AMINOCARBONYL-1,3,4,5-TETRAHYDROBENZ (CD) INDOLE |
1991 |
- Tomas Dzhozef Kress[Us]
- Dehvid Li Vari[Us]
|
RU2034837C1 |
| CEPHALOSPORIN DERIVATIVES AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, PHARMACEUTICAL COMPOSITION |
1992 |
- Robert Dzhon Ternanski[Us]
|
RU2104280C1 |
| PIPERIDINE COMPOUNDS AND PHARMACEUTICAL COMPOSITION SHOWING ACTIVITY AS ANTAGONIST OF OPIOID PERIPHERAL ACTION |
1992 |
- Baddi Judzhin Kantrell[Us]
- Dennis Majkl Tsimmerman[Us]
|
RU2076863C1 |
| PYRAZOLE DERIVATIVES AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS |
1991 |
- Rejmond Frenk Braun[Us]
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- Karen Linn Lobb[Us]
- Dehvid Ehndrju Nil[Us]
- Dzhon Kevin Ril[Us]
|
RU2076100C1 |
