FIELD: organic chemistry. SUBSTANCE: product: derivatives of pyrrole-substituted ureides of the formula (I) $$$ where: m and n are whole numbers 1-3; W - oxygen; B - naphthalene or quinoline ring substituted with 1-3 groups of sulfoacid or 2-deoxy-D-glucose-6-sulfate or 2-deoxy-D-glucose-6-phosphate and their pharmaceutically acceptable salts. Reagent 1: compound of the formula (II) $$$ where: n and B - as indicated above. Reagent 2: compound of the formula: X-C-(W)-X where: W - oxygen; X - halogen, imidazolyl, triazolyl, p-nitrophenoxy- or trichlorophenoxy-group. Reaction conditions: in medium of organic solvent in the presence of the base, at temperature (-10)-(+50) C. Synthesized compounds inhibit angiotensin activity and can be used in medicine. EFFECT: improved method of synthesis. 9 ex, 6 cl, 1 tbl
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