OXAZOLIDINE DERIVATIVES OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS OR ESTERS AND METHOD OF THEIR SYNTHESIS Russian patent published in 1997 - IPC

Abstract RU 2090564 C1

FIELD: chemistry of heterocyclic compounds. SUBSTANCE: product: derivatives of oxazolidine of the formula (I) given in description where: R - C1-C8-alkyl; X - S or O; Y - H or group -A-COOW where: A - C1-C6-alkylene; W - H or C1-C6-alkyl; Ar - aryl group containing 6-10 carbon atoms in ring and possibly substituted with halogen, halide-C1-C4-alkyl, hydroxy-group, C1-C4-alkyl, C1-C4-alkoxy-group, or their salts and esters. Invention proposes method of synthesis of compounds of the formula (I). Synthesized compounds show hypoglycaemic activity. EFFECT: improved method of synthesis. 21 cl, 4 tbl

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RU 2 090 564 C1

Authors

Takasi Fudzita[Jp]

Takao Esioka[Jp]

Sindzi Esioka[Jp]

Tosikhiko Fudzivara[Jp]

Khirojosi Khorikosi[Jp]

Dates

1997-09-20Published

1993-08-30Filed