8-SUBSTITUTED-2-AMINOTETRALINE DERIVATIVES AND METHODS OF PREPARATION THEREOF Russian patent published in 1997 - IPC

Abstract RU 2093507 C1

FIELD: medicine. SUBSTANCE: present invention describes compound of formula (I) in which Z is hydrogen or halogen; Q is CORI or 5- or 6- membered aryl which contains 1 or 2-heteroatoms from N, O and S optionally substituted or condensed wherein R is hydrogen or CI-methyl (cis-configuration); RI is CI-6 alkyl or aromatic ring which contains heteroatoms O or S and is substituted or condensed with optionally substituted benzene ring; R2 is hydrogen or CI-6-alkyl, and R3 is as defined in claim 1, and enantiomers or salts thereof, methods of preparation of said compounds, drugs based thereon, and also method of medical treatment of central nervous system diseases when using said compounds. EFFECT: more efficient preparation method. 16 cl, 1 tbl

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RU 2 093 507 C1

Authors

Nil'S-Ehrik Anden[Se]

Berit Kristina Ehlizabet Baklund Khek[Se]

Anna Lena Marija B'Erk[Se]

Uli Al'F Khaksell[Se]

Sven-Ehrik Khillver[Se]

Ie Liu[Cn]

Eva Sharlotta Mellin[Se]

Eva Marie Persson[Se]

Karl Erk Vallgarda[Se]

Khong Iu[Cn]

Dates

1997-10-20Published

1990-05-23Filed