3-CARBOXALDEHYDE DERIVATIVES OF QUINOLINE Russian patent published in 1997 - IPC

Abstract RU 2097379 C1

FIELD: organic chemistry. SUBSTANCE: invention proposes 3-carboxaldehyde derivatives of quinoline and naphthyridine of the formula (I): where: A, Y, R₁ and R₂ have values given in description. Compounds can be used by injection route. Specific example of these compounds is 1-cyclopropyl-6-fluoro-7-[(1S, 4S)-5-methyl-2,5-diazabicyclo-[2,2,1] -hept-2-yl] -4-oxo-1,4-dihydroquinoline-3-carboxaldehyde. The synthesized compounds show antibacterial activity. EFFECT: improved method of synthesis. 3 cl, 1 tbl

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RU 2 097 379 C1

Authors

Martin R.Dzhefson[Us]

Dates

1997-11-27—Published

1995-01-13—Filed