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2 105 764

(13)

C1

(51)

IPC

(21) (22)

Application

5052881/04, 1992-10-02

(22)

Actual filing date

1992-10-02

(45)

Published

1998-02-27

(72)

Inventor

Diter Binder[At]Jozef Vajnberger[At]

(73)

Holder

Khemish Farmatsojtishe Forshungsgezel'Shaft Mbkh

NEW IMIDAZOLE-5-CARBOXYLIC ACID ACYLALES, METHOD OF PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITION HAVING PROPERTIES OF RECEPTOR ANGIOTENSINE II ANTAGONIST Russian patent published in 1998 - IPC

Abstract RU 2105764 C1

FIELD: pharmaceutical industry. SUBSTANCE: present invention describes new imidazole-5-carboxylic acid acylales of formula I: wherein R1 is optionally unsaturated straight alkyl group having 1 to 6 carbon atoms; R2 is hydrogen, chlorine, bromine, iodine or CF3, and R3 is C1-C10- alkyl, C3-C7- cycloalkyl or benzyl, and pharmaceutically tolerable salts thereof, and method of preparation thereof. The present invention describes pharmaceutical composition in which active ingredient includes imidazole -5-carboxylic acid acylales intended for reducing blood pressure. EFFECT: improved properties of the pharmaceutical composition. 7 cl, 12 dwg, 3 tbl

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RU 2 105 764 C1

Authors

Diter Binder[At]

Jozef Vajnberger[At]

Dates

1998-02-27—Published

1992-10-02—Filed

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