AMINOQUINOLONE DERIVATIVES SUBSTITUTED BY PHENYL OR HETEROAROMATIC GROUP Russian patent published in 1999 - IPC

Abstract RU 2124510 C1

FIELD: medicine. SUBSTANCE: present invention describes novel compounds of formula Ia or Ic: wherein X is hydrogen or halogen; Y is hydrogen or amino group; Z is carboxy; Q is nitrogen or group of formula: wherein R2 is hydrogen, halogen, lower alkoxy or lower alkoxy substituted by one or more halogen atoms; T is methylene group optionally substituted by lower alkyl; R1 is hydrogen, lower alkylene, lower alkynyl, amino group optionally substituted by one lower alkyl, (C3-C6)-cycloalkyl; lower alkoxy, phenyl optionally substituted by one halogen; lower alkyl; R is group (h) or (i). The claimed compounds have anti activity. EFFECT: improved properties of the title compounds. 22 cl, 5 dwg, 110 ex, 31 tbl

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RU 2 124 510 C1

Authors

Tomio Kimura

Tetsusi Katsube

Dates

1999-01-10Published

1993-05-26Filed