BENZOPIPERIDINE DERIVATIVES, BICYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITION BASED ON SAID Russian patent published in 1999 - IPC

FIELD: organic chemistry, pharmacy. SUBSTANCE: invention describes new derivatives of benzopiperidine of the general formula (I) where dotted line means optional double bond where R₅ and R₆ mean independently hydrogen atom, hydroxyl or a group that can be converted in vivo to hydroxyl-group; R¹⁰⁰ means (CH₂)_n where n = 5-10; L means ; G¹ means hydrogen atom, hydrocarbon C₁-C₅-group or divalent group connecting G² and L leading to the formation of 5-7-membered heterocycle and G² means hydrogen atom, hydrocarbon C₁-C₅-group, substituted or unsubstituted divalent group connecting G¹ and L leading to the formation of 5-7-membered heterocycle. Invention describes also pharmaceutical compositions based on compounds of the formula (I). EFFECT: new compounds indicated above. 20 cl, 5 dwg, 25 tbl, 44 ex