FIELD: organic chemistry, medicine, neurology. SUBSTANCE: invention describes the novel derivatives of naphthylamide of the formula (I) 
where R1 is halogen atom, cyano-group; R2 is direct or branched alkyl with 1-6 carbon atoms; R3 is unsubstituted phenyl or phenyl substituted with 1-2 substituents taken among C1-6-alkyl, halogen atom, C1-6-alkoxy- or thio-C1-6-alkoxy-group, 4-pyridinyl-, 3-benzoiso-thiazolyl- or 7-benzo[b]furanyl-group, and their pharmaceutically acceptable acid-additive salts. Compounds of the formula (I) are dopaminergic agents that can be used as antipsychotic drugs for treatment of psychotic patients, for example, with schizophrenia. EFFECT: new compounds indicated above, improved method of treatment, valuable medicinal properties. 4 cl, 1 tbl, 16 ex
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Year |
Author |
Number |
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