FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to derivatives of sulfamic acid of the general formula (I) 
where R, R1, R2, X and Y have values indicated in p. 1 of the invention claim, or their pharmaceutically acceptable salts. Indicated compounds can be an active substance of the pharmaceutical composition that regulates blood plasma cholesterol concentration. Also, invention relates to a method of treatment of patients with hypercholesterolemia or atherosclerosis by administration of indicated compounds or their pharmaceutically acceptable salts at doses 250-3 000 mg/day. EFFECT: enhanced effectiveness of treatment. 15 cl, 2 dwg, 2 tbl, 48 ex
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