COMPOUNDS OF 7-(2-IMIDAZOLINYLAMINO)-QUINOLINE USED AS AGONISTS OF ALPHA-2-ADRENORECEPTORS Russian patent published in 2001 - IPC

Abstract RU 2161967 C2

FIELD: organic chemistry, medicine. SUBSTANCE: invention relates to novel derivatives of quinoline of the general formula (I) where R means unsubstituted C₁-C₃-alkyl or C₂-C₃-alkenyl; R¹ is cyano-group that are agonists of alpha-2-adrenoreceptors and can be used for preparing drugs that are useful for treatment of patients with nose congestion, glaucoma, diarrhea, asthma. Compounds show the expressed antagonistic activity with respect to α-2-adrenoreceptors. EFFECT: new compounds indicated above, enhanced effectiveness in treatment. 9 cl, 1 tbl, 3 ex

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RU 2 161 967 C2

Authors

Tomas Li Kapps

Sofi Eva Bogdan

Dates

2001-01-20—Published

1994-12-15—Filed