DERIVATIVES OF QUINOLINE-2(1H)-ONE, METHODS OF THEIR SYNTHESIS, DRUG AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF Russian patent published in 2001 - IPC

Abstract RU 2167874 C2

FIELD: organic chemistry, pharmacy. SUBSTANCE: invention relates to derivatives of quinoline-2(1H)-one of the general formula (I) where R₁,R₂,R₃, A and n have values indicated in the invention claim and to methods of synthesis of compounds of the formula (I). These compounds show antagonistic activity with respect to serotonin and they are useful for therapeutical aims. EFFECT: improved method of synthesis, valuable medicinal properties. 7 cl, 35 ex

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RU 2 167 874 C2

Authors

Mak Kor Gari

Khornar Kristian

Dellak Zhenev'Ev

Aletrju Mishel'

Dates

2001-05-27—Published

1996-09-12—Filed