METHOD OF PREPARING RACEMIC OR OPTICALLY ACTIVE METHYL (2-HALOGENOPHENYL) (6,7-DIHYDRO-4H-THIENO (3- 2-c) PYRIDIN-5-YL) ACETATES OR SALTS THEREOF Russian patent published in 2001 - IPC

Abstract RU 2172315 C1

FIELD: chemical industry. SUBSTANCE: described is method of preparing racemic or optically active methyl (2-halogenophenyl) (6,7-dihydro-4H- thieno (3,2-c) pyridin-5-yl)acetates of formula VI: or salts thereof by conversion of racemic or optically active compound of formula VII: into compound followed by cyclization of the latter. Said compounds are useful for treatment purposes due to the fact that they inhibit aggregation of thrombocytes. Method makes it possible to increase yield of the desired product and avoid using toxic intermediate compound. EFFECT: improved properties of the title compounds. 5 cl, 22 ex, 2 dwg

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RU 2 172 315 C1

Authors

Bakoni Marija

Chatarine Nad' Marianna

Mol'Nar Leventene

Gajari Antal'

Alatt'Jani Ehdit

Dates

2001-08-20Published

1998-05-11Filed