FIELD: organic synthesis. SUBSTANCE: invention provides novel compounds of general formula C (see description), in which X denotes nitrogen atom, Y group -CH= or CR7 (wherein R7 is lower alkyl or halogen atom), Z group -CH=; R2a optionally substituted amino group or protected amino group, and R3 hydrogen atom or halogen. Pyridone- carboxylic acid derivatives and their salts showing antibacterial activity can be prepared from above-indicated amino compounds. EFFECT: expanded possibilities in synthesis of antibacterial agents. 5 cl, 2 tbl, 102 ex
Title |
Year |
Author |
Number |
DERIVATIVES OF PYRIDONE CARBOXYLIC ACID OR THEIR SALTS AND ANTIBACTERIAL AGENT |
1996 |
- Akira Jazaki
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- Khirotaka Amano
- Norikhiro Khajjasi
- Jasukhiro Kuramoto
|
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DERIVATIVE OF PYRIDONE CARBOXYLIC ACID OR ITS SALT |
1996 |
- Jazaki Akira
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1993 |
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DEHALOGENATED COMPOUNDS, ANTIBACTERIAL AGENT AND THERAPEUTIC AGENT BASED ON THEREOF, METHOD FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT, USING DEHALOGENATED COMPOUNDS FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT |
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