LIDINE-1-YL-ACETYLAMINO)-3-PHENYLPROPIONIC ACID ETHYL ESTER SALTS, METHOD OF THEIR SYNTHESIS AND PHARMACEUTICAL COMPOSITION BASED ON THEREOF Russian patent published in 2001 - IPC

Abstract RU 2174119 C2

FIELD: organic chemistry, chemical technology, pharmacy. SUBSTANCE: invention relates to compounds of the formula (I) in all stereoisomeric forms and their mixtures in any ratios where HB means maleic acid, to method of synthesis of compounds of the formula (I) that involves anionic exchange of compounds of the formula (II) with maleic acid and/or maleates. Invention relates to also the pharmaceutical composition showing inhibitory effect on platelet aggregation or suppressing effect with respect of thrombosis. Therefore, compounds of the general formula (I) can be used as medicinal agents for prophylaxis of diseases associated with cardiovascular injuries. EFFECT: improved method of synthesis, valuable medicinal properties of compounds. 10 cl, 5 ex

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RU 2 174 119 C2

Authors

Khans Ul'Rikh Shtil'Ts

Gerkhard Bekk

Manfred Radau

Dates

2001-09-27Published

1997-06-05Filed