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2 188 827

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(51)

IPC

(21) (22)

Application

2000124761/04, 2000-09-28

(24)

Start date

2000-09-28

(22)

Actual filing date

2000-09-28

(45)

Published

2002-09-10

(72)

Inventor

Kaneko TakusiMaklaflin Robert Uill'JamMakmillen Uill'Jam TomasRipin Dehvid Garol'D BraunVanderplas Brajan Klement

(73)

Holder

Pfajzer Prodakts Ink.

CARBAMATE KETOLIDE ANTIBIOTICS, METHODS OF THEIR SYNTHESIS, INTERMEDIATE COMPOUNDS Russian patent published in 2002 - IPC

Abstract RU 2188827 C2

FIELD: organic chemistry, antibiotics. SUBSTANCE: invention relates to a method of synthesis of macrolide antibiotic characterized by the formula (15) where substitutes R¹, R², R³, R⁴, R⁵ have values indicated in the invention description. These antibiotics can be used as antibacterial and antiprotozoan agents for mammals including humans, fishes and birds. Invention presents also novel compounds that can be synthesized using the synthesis of a macrolide antibiotic. EFFECT: improved methods of synthesis. 28 cl

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RU 2 188 827 C2

Authors

Kaneko Takusi

Maklaflin Robert Uill'Jam

Makmillen Uill'Jam Tomas

Ripin Dehvid Garol'D Braun

Vanderplas Brajan Klement

Dates

2002-09-10—Published

2000-09-28—Filed